Dr. Jürgen Einsiedel

Lehrstuhl für Pharmazeutische Chemie

Structure-based discovery of CFTR potentiators and inhibitors (2024) Liu F, Kaplan AL, Levring J, Einsiedel J, Tiedt S, Distler K, Omattage NS, et al. Journal article The small molecule activator S3969 stimulates the epithelial sodium channel by interacting with a specific binding pocket in the channel's β-subunit (2024) Sure F, Einsiedel J, Gmeiner P, Duchstein P, Zahn D, Korbmacher C, Ilyaskin A Journal article Development of disulfide-functionalized peptides covalently binding G protein-coupled receptors (2022) Einsiedel J, Schmidt M, Hübner H, Gmeiner P Journal article Sensitization to amphetamine psychostimulant effect: A key role for ventral tegmental area neurotensin type 2 receptors and MAP kinase pathway (2021) Voyer D, Einsiedel J, Gmeiner P, Lévesque D, Rompré PP Journal article Structure-based exploration of an allosteric binding pocket in the NTS1 receptor using bitopic NT(8-13) derivatives and molecular dynamics simulations (2019) Kling R, Burchardt C, Einsiedel J, Hübner H, Gmeiner P Journal article NTS2-selective neurotensin mimetics with tetrahydrofuran amino acids (2017) Simeth NA, Bause M, Dobmeier M, Kling R, Lachmann D, Hübner H, Einsiedel J, et al. Journal article, Original article Theranostic Value of Multimers: Lessons Learned from Trimerization of Neurotensin Receptor Ligands and Other Targeting Vectors (2017) Maschauer S, Einsiedel J, Reich D, Hübner H, Gmeiner P, Wester HJ, Prante O, Notni J Journal article, Original article Mimicking of Arginine by Functionalized N(ω)-Carbamoylated Arginine As a New Broadly Applicable Approach to Labeled Bioactive Peptides: High Affinity Angiotensin, Neuropeptide Y, Neuropeptide FF, and Neurotensin Receptor Ligands As Examples. (2016) Keller M, Kuhn KK, Einsiedel J, Hübner H, Biselli S, Mollereau C, Wifling D, et al. Journal article, Original article Discovery and Characterization of Biased Allosteric Agonists of the Chemokine Receptor CXCR3. (2016) Lampros M, Brox R, Frank T, Poklukar G, Palmisano R, Waibel R, Einsiedel J, et al. Journal article 18F- and 68Ga-Labeled Neurotensin Peptides for PET Imaging of Neurotensin Receptor 1 (2016) Maschauer S, Einsiedel J, Hübner H, Gmeiner P, Prante O Journal article, Original article