Dr. Harald Hübner

Lehrstuhl für Pharmazeutische Chemie

Rationally Based Efficacy Tuning of Selective Dopamine D4 Receptor Ligands Leading to the Complete Antagonist 2-[4-(4-Chlorophenyl)piperazin-1-ylmethyl]pyrazolo[1,5-a]pyridine (FAUC 213) (2001) Utz W, Löber S, Gmeiner P, Hübner H Journal article Planar Chiral Indoles: Synthesis and Biological Effects of the Enantiomers (2001) Gmeiner P, Hübner H Journal article Dopaminergic 7-Aminotetrahydroindolizines: Ex-Chiral Pool Synthesis and Preferential D3 Receptor Binding (2001) Gmeiner P, Hübner H Journal article Benzamide Bioisosteres Incorporating Dihydroheteroazole Substructures: EPC Synthesis and SAR Leading to a Selective Dopamine D4 Receptor Partial Agonist (FAUC 179) (2001) Gmeiner P, Einsiedel J, Hübner H Journal article Phenyloxazoles and Phenylthiazoles as Benzamide Bioisosteres: Synthesis and Dopamine Receptor Binding Profiles (2000) Gmeiner P, Einsiedel J, Hübner H Journal article Cyanoindole Derivatives as Highly Selective Dopamine D4 Receptor Partial Agonists: Solid-Phase Synthesis, Binding Assays, and Functional Experiments (2000) Gmeiner P, Hübner H Journal article Conjugated Enynes as Nonaromatic Catechol Bioisosteres: Synthesis, Binding Experiments and Computational Studies of Novel Dopamine Receptor Agonists Recognizing Preferentially the D3 Subtype (2000) Utz W, Gmeiner P, Hübner H Journal article Azepino- and Diazepinoindoles: Synthesis and Dopamine Receptor Binding Profiles (2000) Gmeiner P, Hübner H Journal article Piperidinylpyrroles: Design, Synthesis and Binding Properties of Novel and Selective Dopamine D4 Receptor Ligands (1999) Hübner H, Gmeiner P Journal article Enantio- and Diastereocontrolled Dopamine D1, D2, D3 and D4 Receptor Binding of N-(3-Pyrrolidinylmethyl)benzamides Synthesized from Aspartic Acid (1999) Hübner H, Gmeiner P Journal article