Prof. Dr. Peter Gmeiner

Lehrstuhl für Pharmazeutische Chemie

Short and Efficient Synthesis of Homo-Freidinger Lactams: An Olefin Metathesis Approach Towards Conformationally Restricted ß-Amino Acid Analogues (2002) Gmeiner P Journal article Comparative molecular field analysis of dopamine D4 receptor antagonists including 3-[4-(4-chlorophenyl)piperazin-1-ylmethyl]pyrazolo[1,5-a]pyridine (FAUC 113), 3-[4-(4-chlorophenyl)piperazin-1-ylmethyl]-1H-pyrrolo-[2,3-b]pyridine (L-745,870), and clozapine. (2001) Lanig H, Utz W, Gmeiner P Journal article, Original article Comparative Molecular Field Analysis of Dopamine D4 Receptor Antagonists Including 3-[4-(4-Chlorophenyl)piperazin-1-ylmethyl]pyrazolo[1,5-a]pyridine (FAUC 113), 3-[4-(4-Chlorophenyl)piperazin-1-ylmethyl]-1H-pyrrolo[2,3-b]pyridine (L-745,870), and Clozapine (2001) Lanig H, Utz W, Gmeiner P, Lanig H Journal article, Original article Synthesis and in vitro Evaluation of Iodine Labelled Pyrazolo[1,5-a]pyridines as Highly Selective Dopamine D4 Receptor Ligands (2001) Löber S, Gmeiner P, Hübner H Journal article Rationally Based Efficacy Tuning of Selective Dopamine D4 Receptor Ligands Leading to the Complete Antagonist 2-[4-(4-Chlorophenyl)piperazin-1-ylmethyl]pyrazolo[1,5-a]pyridine (FAUC 213) (2001) Utz W, Löber S, Gmeiner P, Hübner H Journal article Planar Chiral Indoles: Synthesis and Biological Effects of the Enantiomers (2001) Gmeiner P, Hübner H Journal article Indoloparacyclophanes: Synthesis and Dopamine Receptor Binding of a Novel Arylbioisostere (2001) Waibel R, Gmeiner P Journal article Dopaminergic 7-Aminotetrahydroindolizines: Ex-Chiral Pool Synthesis and Preferential D3 Receptor Binding (2001) Gmeiner P, Hübner H Journal article Diethoxymethyl Protected Pyrroles: Synthesis and Regioselective Transformations (2001) Gmeiner P Journal article Benzamide Bioisosteres Incorporating Dihydroheteroazole Substructures: EPC Synthesis and SAR Leading to a Selective Dopamine D4 Receptor Partial Agonist (FAUC 179) (2001) Gmeiner P, Einsiedel J, Hübner H Journal article