Journal of Medicinal Chemistry
Journal Abbreviation: J MED CHEM
ISSN: 0022-2623
eISSN: 1520-4804
Publisher: American Chemical Society
Publications (68)
Dual-Acting Cholinesterase-Human Cannabinoid Receptor 2 Ligands Show Pronounced Neuroprotection in Vitro and Overadditive and Disease-Modifying Neuroprotective Effects in Vivo (2019)
Scheiner M, Dolles D, Gunesch S, Hoffmann M, Nabissi M, Marinelli O, Naldi M, et al.
Journal article, Original article
A New Fluorogenic Small-Molecule Labeling Tool for Surface Diffusion Analysis and Advanced Fluorescence Imaging of β-Site Amyloid Precursor Protein-Cleaving Enzyme 1 Based on Silicone Rhodamine: SiR-BACE1 (2018)
Karch S, Broichhagen J, Schneider J, Boening D, Hartmann S, Schmid B, Tripal P, et al.
Journal article
Structure-Based Design and Discovery of New M-2 Receptor Agonists (2017)
Fish I, Stößel A, Eitel K, Valant C, Albold S, Hübner H, Möller D, et al.
Journal article, Original article
Hydroxy-Substituted Heteroarylpiperazines: Novel Scaffolds for beta-Arrestin-Biased D2R Agonists (2017)
Männel B, Dengler D, Shonberg J, Hübner H, Möller D, Gmeiner P
Journal article, Original article
Radiolabeled Dibenzodiazepinone-Type Antagonists Give Evidence of Dualsteric Binding at the M-2 Muscarinic Acetylcholine Receptor (2017)
Pegoli A, She X, Wifling D, Hübner H, Bernhardt G, Gmeiner P, Keller M
Journal article, Original article
Discovery of G Protein-Biased Dopaminergics with a Pyrazolo[1,5-a]pyridine Substructure (2017)
Möller D, Banerjee A, Uzuneser T, Skultety M, Huth T, Plouffe B, Hübner H, et al.
Journal article, Original article
Design, Synthesis, and Biological Evaluation of Small, High-Affinity Siglec-7 Ligands: Toward Novel Inhibitors of Cancer Immune Evasion (2017)
Prescher H, Frank M, Guetgemann S, Kuhfeldt E, Schweizer A, Nitschke L, Watzl C, Brossmer R
Journal article
Mimicking of Arginine by Functionalized N(ω)-Carbamoylated Arginine As a New Broadly Applicable Approach to Labeled Bioactive Peptides: High Affinity Angiotensin, Neuropeptide Y, Neuropeptide FF, and Neurotensin Receptor Ligands As Examples. (2016)
Keller M, Kuhn KK, Einsiedel J, Hübner H, Biselli S, Mollereau C, Wifling D, et al.
Journal article, Original article
Discovery and Characterization of Biased Allosteric Agonists of the Chemokine Receptor CXCR3. (2016)
Lampros M, Brox R, Frank T, Poklukar G, Palmisano R, Waibel R, Einsiedel J, et al.
Journal article
18F- and 68Ga-Labeled Neurotensin Peptides for PET Imaging of Neurotensin Receptor 1 (2016)
Maschauer S, Einsiedel J, Hübner H, Gmeiner P, Prante O
Journal article, Original article