Journal of Medicinal Chemistry
Journal Abbreviation: J MED CHEM
ISSN: 0022-2623
eISSN: 1520-4804
Publisher: American Chemical Society
Publications (63)
Regiospecific Introduction of Halogens on the 2-Aminobiphenyl Subunit Leading to Highly Potent and Selective M3 Muscarinic Acetylcholine Receptor Antagonists and Weak Inverse Agonists (2020)
Fischer O, Hofmann J, Rampp H, Kaindl J, Pratsch G, Bartuschat A, Taudte V, et al.
Journal article
Investigation of Inactive-State κ Opioid Receptor Homodimerization via Single-Molecule Microscopy Using New Antagonistic Fluorescent Probes (2020)
Drakopoulos A, Koszegi Z, Lanoiselée Y, Hübner H, Gmeiner P, Calebiro D, Decker M
Journal article
Conjugation of Short Peptides to Dibenzodiazepinone-Type Muscarinic Acetylcholine Receptor Ligands Determines M2R Selectivity (2019)
Pegoli A, Wifling D, Gruber CG, She X, Hübner H, Bernhardt G, Gmeiner P, Keller M
Journal article
Hybridization of β-Adrenergic Agonists and Antagonists Confers G Protein Bias (2019)
Stanek M, Picard LP, Schmidt M, Kaindl J, Hübner H, Bouvier M, Weikert D, Gmeiner P
Journal article
Benzyl Phenylsemicarbazides: A Chemistry-Driven Approach Leading to G Protein-Biased Dopamine D4 Receptor Agonists with High Subtype Selectivity (2019)
Pirzer A, Lasch R, Friedrich H, Hübner H, Gmeiner P, Heinrich M
Journal article, Original article
Dual-Acting Cholinesterase-Human Cannabinoid Receptor 2 Ligands Show Pronounced Neuroprotection in Vitro and Overadditive and Disease-Modifying Neuroprotective Effects in Vivo (2019)
Scheiner M, Dolles D, Gunesch S, Hoffmann M, Nabissi M, Marinelli O, Naldi M, et al.
Journal article, Original article
A New Fluorogenic Small-Molecule Labeling Tool for Surface Diffusion Analysis and Advanced Fluorescence Imaging of β-Site Amyloid Precursor Protein-Cleaving Enzyme 1 Based on Silicone Rhodamine: SiR-BACE1 (2018)
Karch S, Broichhagen J, Schneider J, Boening D, Hartmann S, Schmid B, Tripal P, et al.
Journal article
Structure-Based Design and Discovery of New M-2 Receptor Agonists (2017)
Fish I, Stößel A, Eitel K, Valant C, Albold S, Hübner H, Möller D, et al.
Journal article, Original article
Hydroxy-Substituted Heteroarylpiperazines: Novel Scaffolds for beta-Arrestin-Biased D2R Agonists (2017)
Männel B, Dengler D, Shonberg J, Hübner H, Möller D, Gmeiner P
Journal article, Original article
Radiolabeled Dibenzodiazepinone-Type Antagonists Give Evidence of Dualsteric Binding at the M-2 Muscarinic Acetylcholine Receptor (2017)
Pegoli A, She X, Wifling D, Hübner H, Bernhardt G, Gmeiner P, Keller M
Journal article, Original article