Dr. Jürgen Einsiedel



Organisation


Lehrstuhl für Pharmazeutische Chemie


Publications (Download BibTeX)

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Kling, R., Burchardt, C., Einsiedel, J., Hübner, H., & Gmeiner, P. (2019). Structure-based exploration of an allosteric binding pocket in the NTS1 receptor using bitopic NT(8-13) derivatives and molecular dynamics simulations. Journal of Molecular Modeling, 25(7). https://dx.doi.org/10.1007/s00894-019-4064-x
Simeth, N.A., Bause, M., Dobmeier, M., Kling, R., Lachmann, D., Hübner, H.,... Koenig, B. (2017). NTS2-selective neurotensin mimetics with tetrahydrofuran amino acids. Bioorganic & Medicinal Chemistry, 25(1), 350-359. https://dx.doi.org/10.1016/j.bmc.2016.10.039
Maschauer, S., Einsiedel, J., Reich, D., Hübner, H., Gmeiner, P., Wester, H.J.,... Notni, J. (2017). Theranostic Value of Multimers: Lessons Learned from Trimerization of Neurotensin Receptor Ligands and Other Targeting Vectors. Pharmaceuticals, 10(1), 29. https://dx.doi.org/10.3390/ph10010029
Maschauer, S., Einsiedel, J., Hübner, H., Gmeiner, P., & Prante, O. (2016). 18F- and 68Ga-Labeled Neurotensin Peptides for PET Imaging of Neurotensin Receptor 1. Journal of Medicinal Chemistry, 59, 6480-6492. https://dx.doi.org/10.1021/acs.jmedchem.6b00675
Lampros, M., Brox, R., Frank, T., Poklukar, G., Palmisano, R., Waibel, R.,... Tschammer, N. (2016). Discovery and Characterization of Biased Allosteric Agonists of the Chemokine Receptor CXCR3. Journal of medicinal chemistry, 59(5), 2222-43. https://dx.doi.org/10.1021/acs.jmedchem.5b01965
Keller, M., Kuhn, K.K., Einsiedel, J., Hübner, H., Biselli, S., Mollereau, C.,... Buschauer, A. (2016). Mimicking of Arginine by Functionalized N(ω)-Carbamoylated Arginine As a New Broadly Applicable Approach to Labeled Bioactive Peptides: High Affinity Angiotensin, Neuropeptide Y, Neuropeptide FF, and Neurotensin Receptor Ligands As Examples. Journal of medicinal chemistry, 59(5), 1925-45. https://dx.doi.org/10.1021/acs.jmedchem.5b01495
Maschauer, S., Greff, C., Einsiedel, J., Ott, J., Tripal, P., Hübner, H.,... Prante, O. (2015). Improved radiosynthesis and preliminary in vivo evaluation of a 18F-labeled glycopeptide-peptoid hybrid for PET imaging of neurotensin receptor 2. Bioorganic & Medicinal Chemistry, 23, 4026-4033. https://dx.doi.org/10.1016/j.bmc.2015.01.053
Hutterer, C., Niemann, I., Milbradt, J., Fröhlich, T., Reiter, C., Kadioglu, O.,... Marschall, M. (2015). The broad-spectrum antiinfective drug artesunate interferes with the canonical nuclear factor kappa B (NF-κB) pathway by targeting RelA/p65. Antiviral Research, 124, 101-109. https://dx.doi.org/10.1016/j.antiviral.2015.10.003
Haubner, R., Maschauer, S., Einsiedel, J., Eder, I.E., Rangger, C., Gmeiner, P.,... Prante, O. (2014). H-CRRETAWAC-OH, a Lead Structure for the Development of Radiotracer Targeting Integrin Alpha5Beta1? BioMed Research International, 2014, 243185. https://dx.doi.org/10.1155/2014/243185
Maschauer, S., Ruckdeschel, T., Tripal, P., Haubner, R., Einsiedel, J., Hübner, H.,... Prante, O. (2014). In vivo monitoring of the antiangiogenic effect of neurotensin receptor-mediated radiotherapy by small-animal positron emission tomography: A pilot study. Pharmaceuticals, 7(4), 464-481. https://dx.doi.org/10.3390/ph7040464

Last updated on 2016-05-05 at 05:13