Planar Chiral Indoles: Synthesis and Biological Effects of the Enantiomers

Gmeiner P, Hübner H (2001)

Publication Type: Journal article

Publication year: 2001

Journal

Tetrahedron-Asymmetry Elsevier

Publisher: Elsevier

Book Volume: 12

Pages Range: 3205-3208

DOI: 10.1016/S0957-4166(01)00558-4

Abstract

The paracyclophanyl triflates (R)-4 and (S)-4, which were obtained from racemic precursors through enzymatic-kinetic resolution, could be employed as key intermediates for the synthesis of planar chiral [2.2](4,7)indoloparacyclophanes. Subjecting the double-layered test compounds (R)-8 and (S)-8 to in vitro ligand-binding experiments displayed stereoselective receptor recognition. © 2002 Elsevier Science Ltd. All rights reserved.

Authors with CRIS profile

Peter Gmeiner Lehrstuhl für Pharmazeutische Chemie Harald Hübner Lehrstuhl für Pharmazeutische Chemie

How to cite

APA:

Gmeiner, P., & Hübner, H. (2001). Planar Chiral Indoles: Synthesis and Biological Effects of the Enantiomers. Tetrahedron-Asymmetry, 12, 3205-3208. https://doi.org/10.1016/S0957-4166(01)00558-4

MLA:

Gmeiner, Peter, and Harald Hübner. "Planar Chiral Indoles: Synthesis and Biological Effects of the Enantiomers." Tetrahedron-Asymmetry 12 (2001): 3205-3208.

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