Synthesis and Stereochemistry of Oxazolo[4',5':1,2]benz[5,4,3-c,d]indole Derivatives as Intermediates on the Way to a Selective Dopamine Autoreceptor Agonist

Gmeiner P (1996)


Publication Type: Journal article

Publication year: 1996

Journal

Publisher: Wiley-Blackwell

Book Volume: 33

Pages Range: 481-483

Abstract

An expedient and practical variant of the synthesis of the selective dopamine autoreceptor agonist 5 from the benzindolone 1 is described. The reaction sequence includes a two-fold epimerization at the α-position of the lactam function. The structure of the intermediate 9a was confirmed by X-ray structure analysis.

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How to cite

APA:

Gmeiner, P. (1996). Synthesis and Stereochemistry of Oxazolo[4',5':1,2]benz[5,4,3-c,d]indole Derivatives as Intermediates on the Way to a Selective Dopamine Autoreceptor Agonist. Journal of Heterocyclic Chemistry, 33, 481-483.

MLA:

Gmeiner, Peter. "Synthesis and Stereochemistry of Oxazolo[4',5':1,2]benz[5,4,3-c,d]indole Derivatives as Intermediates on the Way to a Selective Dopamine Autoreceptor Agonist." Journal of Heterocyclic Chemistry 33 (1996): 481-483.

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