apl. Prof. Dr. Jörg König

Medizinische Fakultät Lehrstuhl für Klinische Pharmakologie und Klinische Toxikologie

Heteroaryl derivatives of suvorexant as OX1R selective PET ligand candidates: Cu-mediated 18F-fluorination of boroxines, in vitro and initial in vivo evaluation (2024) Bolik KV, Hellmann J, Maschauer S, Neu E, Einsiedel J, Riss P, Vogg N, et al. Journal article Transport of aromatic amino acids l-tryptophan, l-tyrosine, and l-phenylalanine by the organic anion transporting polypeptide (OATP) 3A1 (2024) Surrer D, Schüsser S, König J, Fromm M, Geßner A Journal article New Biomarkers for Renal Transporter-Mediated Drug–Drug Interactions: Metabolomic Effects of Cimetidine, Probenecid, Verapamil, and Rifampin in Humans (2024) Geßner A, König J, Wenisch P, Heinrich M, Stopfer P, Fromm M, Müller F Journal article A Metabolomic Analysis of Sensitivity and Specificity of 23 Previously Proposed Biomarkers for Renal Transporter-Mediated Drug-Drug Interactions (2023) Geßner A, Müller F, Wenisch P, Heinrich M, König J, Stopfer P, Fromm M Journal article Novel drug transporter substrates identification: An innovative approach based on metabolomic profiling, in silico ligand screening and biological validation (2023) Nies AT, König J, Leuthold P, Damme K, Winter S, Haag M, Masuda S, et al. Journal article Transcriptional Regulation of Liver-Type OATP1B3 (Lt-OATP1B3) and Cancer-Type OATP1B3 (Ct-OATP1B3) Studied in Hepatocyte-Derived and Colon Cancer-Derived Cell Lines (2023) Haberkorn B, Löwen D, Meier L, Fromm M, König J Journal article Exploring Structural Determinants of Bias among D4 Subtype-Selective Dopamine Receptor Agonists (2023) Graßl F, Bock L, Huete-Huerta González Á, Schiller M, Gmeiner P, König J, Fromm M, et al. Journal article Cancer-Type Organic Anion Transporting Polypeptide 1B3 Is Localized in Lysosomes and Mediates Resistance against Kinase Inhibitors (2022) Haberkorn B, Oswald S, Kehl N, Geßner A, Taudte V, Dobert J, Zunke F, et al. Journal article Cell-Specific Transport and Thyroid Hormone Receptor Isoform Selectivity Account for Hepatocyte-Targeted Thyromimetic Action of MGL-3196 (2022) Hönes GS, Sivakumar RG, Hoppe C, König J, Führer D, Moeller LC Journal article A Novel and Cross-Species Active Mammalian INDY (NaCT) Inhibitor Ameliorates Hepatic Steatosis in Mice with Diet-Induced Obesity (2022) Zahn G, Willmes DM, El-Agroudy NN, Yarnold C, Jarjes-Pike R, Schaertl S, Schreiter K, et al. Journal article