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Dr. Dorothée Weikert
Orcid ID:
0000-0003-2259-9002
List of publications:
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Lehrstuhl für Pharmazeutische Chemie
Publications
(37)
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Discovery of Novel Nonpeptidic PAR2 Ligands (2020)
Klösel I, Schmidt M, Kaindl J, Hübner H, Weikert D, Gmeiner P
Journal article
Rational design of agonists for bitter taste receptor TAS2R14: from modeling to bench and back (2020)
Di Pizio A, Waterloo L, Brox R, Löber S, Weikert D, Behrens M, Gmeiner P, Niv MY
Journal article
Differential allosteric modulation within dopamine D2R - neurotensin NTS1R and D2R - serotonin 5-HT2AR receptor complexes gives bias to intracellular calcium signalling. (2019)
Plach M, Schäfer T, Borroto-Escuela DO, Weikert D, Gmeiner P, Fuxe K, Friedland K
Journal article, Original article
Hybridization of β-Adrenergic Agonists and Antagonists Confers G Protein Bias (2019)
Stanek M, Picard LP, Schmidt M, Kaindl J, Hübner H, Bouvier M, Weikert D, Gmeiner P
Journal article
Structure-Based Design and Discovery of New M-2 Receptor Agonists (2017)
Fish I, Stößel A, Eitel K, Valant C, Albold S, Hübner H, Möller D, et al.
Journal article, Original article
beta-Arrestin biased dopamine D2 receptor partial agonists: Synthesis and pharmacological evaluation (2017)
Männel B, Hübner H, Möller D, Gmeiner P
Journal article, Original article
Structure-Guided Screening for Functionally Selective D-2 Dopamine Receptor Ligands from a Virtual Chemical Library (2017)
Männel B, Jaiteh M, Zeifinan A, Randakova A, Möller D, Hübner H, Gmeiner P, Carlsson J
Journal article, Original article
Hydroxy-Substituted Heteroarylpiperazines: Novel Scaffolds for beta-Arrestin-Biased D2R Agonists (2017)
Männel B, Dengler D, Shonberg J, Hübner H, Möller D, Gmeiner P
Journal article, Original article
Discovery of G Protein-Biased Dopaminergics with a Pyrazolo[1,5-a]pyridine Substructure (2017)
Möller D, Banerjee A, Uzuneser T, Skultety M, Huth T, Plouffe B, Hübner H, et al.
Journal article, Original article
Visualization of ligand-induced dopamine D2S and D2L receptor internalization by TIRF microscopy (2017)
Tabor A, Möller D, Hübner H, Kornhuber J, Gmeiner P
Journal article, Original article
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