Lehrstuhl für Pharmazeutische Chemie

Heteroaryl derivatives of suvorexant as OX1R selective PET ligand candidates: Cu-mediated 18F-fluorination of boroxines, in vitro and initial in vivo evaluation (2024) Bolik KV, Hellmann J, Maschauer S, Neu E, Einsiedel J, Riss P, Vogg N, et al. Journal article Synthesis, biological evaluation, and molecular docking of novel 1,3,4-substituted-thiadiazole derivatives as potential anticancer agent (2024) Shaikh SA, Wakchaure S, Labhade SR, Kale RR, Alavala RR, Chobe SS, Jain KS, et al. Journal article Identification of novel inhibitors of the transcriptional coactivator MRTF-A for HCC therapy (2024) Franz M, Wenisch P, Wohlleben P, Rupprecht L, Chubanov V, Gudermann T, Kyheröinen S, et al. Journal article Design, Synthesis, and Characterization of New δ Opioid Receptor-Selective Fluorescent Probes and Applications in Single-Molecule Microscopy of Wild-Type Receptors (2024) Drakopoulos A, Koszegi Z, Seier K, Hübner H, Maurel D, Sounier R, Granier S, et al. Journal article Structure-based discovery of CFTR potentiators and inhibitors (2024) Liu F, Kaplan AL, Levring J, Einsiedel J, Tiedt S, Distler K, Omattage NS, et al. Journal article Development and Initial Characterization of the First 18F-CXCR2-Targeting Radiotracer for PET Imaging of Neutrophils (2024) Spatz P, Chen X, Reichau K, Huber M, Mühlig S, Matsusaka Y, Schiedel M, et al. Journal article The small molecule activator S3969 stimulates the epithelial sodium channel by interacting with a specific binding pocket in the channel's β-subunit (2024) Sure F, Einsiedel J, Gmeiner P, Duchstein P, Zahn D, Korbmacher C, Ilyaskin A Journal article Structural and functional characterization of the endogenous agonist for orphan receptor GPR3 (2024) Chen G, Staffen N, Wu Z, Xu X, Pan J, Inoue A, Shi T, et al. Journal article, Letter New fluorogenic triacylglycerols as sensors for dynamic measurement of lipid oxidation (2024) Handke M, Beierlein F, Imhof P, Schiedel M, Hammann S Journal article Dually Labeled Neurotensin NTS1R Ligands for Probing Radiochemical and Fluorescence-Based Binding Assays (2024) Ertl FJ, Kopanchuk S, Dijon NC, Veikšina S, Tahk MJ, Laasfeld T, Schettler F, et al. Journal article