Journal of Medicinal Chemistry
Journal Abbreviation: J MED CHEM
ISSN: 0022-2623
eISSN: 1520-4804
Publisher: American Chemical Society
Publications (73)
1,1′-Disubstituted ferrocenes as molecular hinges in mono- and bivalent dopamine receptor ligands (2009)
Huber D, Hübner H, Gmeiner P
Journal article, Original article
Dopamine D2, D3, and D4 selective phenylpiperazines as molecular probes to explore the origins of subtype specific receptor binding. (2009)
Ehrlich K, Götz A, Bollinger S, Tschammer N, Bettinetti L, Härterich S, Hübner H, et al.
Journal article, Original article
Identification of new functional inhibitors of acid sphingomyelinase using a structure-property-activity relation model (2008)
Kornhuber J, Tripal P, Reichel M, Terfloth L, Bleich S, Wiftfang J, Gulbins E
Journal article
Novel D3 Selective Dopaminergics Incorporating Enyne Units as Nonaromatic Catechol Bioisosteres: Synthesis, Bioactivity, and Mutagenesis Studies (2008)
Doerfler M, Tschammer N, Hamperl K, Hübner H, Gmeiner P
Journal article
Synthesis, Radiofluorination and In Vitro Evaluation of Pyrazolo[1,5-a]pyridine Based Dopamine D4 Receptor Ligands: Discovery of an Inverse Agonist Radioligand for PET (2008)
Prante O, Tietze R, Hocke C, Löber S, Hübner H, Kuwert T, Gmeiner P
Journal article
Structure-Selectivity Investigations of D2-like Receptor Ligands by CoMFA and CoMSIA Guiding the Discovery of D3 Selective PET Radioligands (2007)
Utz W, Prante O, Hübner H, Kuwert T, Gmeiner P
Journal article
Structural changes and binding characteristics of the tetracycline-repressor binding site on induction (2006)
Lanig H, Othersen O, Seidel U, Beierlein F, Exner T, Clark T
Journal article
Fancy Bioisosteres: Novel Paracyclophane Derivatives as Super-Affinity Dopamine D3 Receptor Antagonists (2006)
Gmeiner P, Hübner H
Journal article
A Chimeric Ligand Approach Leading to Potent Antiprion Active Acridine Derivatives: Design, Synthesis and Biological Investigations (2006)
Löber S, Gmeiner P
Journal article
2-[(4-Phenylpiperazin-1-yl)methyl]imidazo(di)azines as Selective D4-Ligands. Induction of Penile Erection by 2-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]imidazo[1,2-a]pyridine (PIP3EA), a Potent and Selective D4 Partial Agonist (2006)
Gmeiner P, Hübner H
Journal article