Microwave-assisted rapid one-pot synthesis of fused and non-fused indoles and 5-[18F]fluoroindoles from phenylazocarboxylates

Krüll J, Hubert A, Nebel N, Prante O, Heinrich M (2017)


Publication Type: Journal article

Publication year: 2017

Journal

DOI: 10.1002/chem.201703890

Abstract

Substituted indoles can be prepared from phenylazo-carboxylates through a rapid one-pot sequence featuring a microwave-assisted Fischer indole synthesis as key step. As the phenylazocarboxylates may beforehand be modified by mild nucleophilic aromatic substitution, including the introduction of [18F]fluoride, the overall strategy offers an attractive new access to 5-[18F]fluoroindoles.

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How to cite

APA:

Krüll, J., Hubert, A., Nebel, N., Prante, O., & Heinrich, M. (2017). Microwave-assisted rapid one-pot synthesis of fused and non-fused indoles and 5-[18F]fluoroindoles from phenylazocarboxylates. Chemistry - A European Journal. https://dx.doi.org/10.1002/chem.201703890

MLA:

Krüll, Jasmin, et al. "Microwave-assisted rapid one-pot synthesis of fused and non-fused indoles and 5-[18F]fluoroindoles from phenylazocarboxylates." Chemistry - A European Journal (2017).

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