Efficient synthesis of heterocyclic neurotensin receptor ligands by microwave-assisted aminocarbonylation

Lang C, Gmeiner P (2013)

Publication Language: English

Publication Type: Journal article, Original article

Publication year: 2013

Journal

Synthesis-Stuttgart Thieme Publishing / Georg Thieme Verlag

Original Authors: Lang C., Gmeiner P.

Publisher: Thieme Publishing / Georg Thieme Verlag

Book Volume: 45

Pages Range: 2474-2480

Journal Issue: 17

DOI: 10.1055/s-0033-1338497

Abstract

Marking the heterocyclic neurotensin receptor antagonist SR142948A as a lead compound, the development of an efficient and a practical synthetic route to heterocyclic aryl carboxamides is reported. Thus, a highly efficient and flexible access to these carboxamides was elaborated by taking advantage of microwave-assisted aminocarbonylation reaction mediated by Mo(CO), Herrmann's palladacycle, [(t-Bu)PH]BF, and DBU. © 2013 Georg Thieme Verlag Stuttgart New York.

Authors with CRIS profile

Christopher Lang Lehrstuhl für Pharmazeutische Chemie Peter Gmeiner Lehrstuhl für Pharmazeutische Chemie

Additional Organisation(s)

Emil-Fischer-Zentrum (Emil Fischer Center)

How to cite

APA:

Lang, C., & Gmeiner, P. (2013). Efficient synthesis of heterocyclic neurotensin receptor ligands by microwave-assisted aminocarbonylation. Synthesis-Stuttgart, 45(17), 2474-2480. https://doi.org/10.1055/s-0033-1338497

MLA:

Lang, Christopher, and Peter Gmeiner. "Efficient synthesis of heterocyclic neurotensin receptor ligands by microwave-assisted aminocarbonylation." Synthesis-Stuttgart 45.17 (2013): 2474-2480.

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