Dr. Harald Hübner



Organisation


Lehrstuhl für Pharmazeutische Chemie


Publications (Download BibTeX)

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Xu, J., Hu, Y., Kaindl, J., Risel, P., Hübner, H., Maeda, S.,... Kobilka, B.K. (2019). Conformational Complexity and Dynamics in a Muscarinic Receptor Revealed by NMR Spectroscopy. Molecular Cell, 75(1), 53-65.e7. https://dx.doi.org/10.1016/j.molcel.2019.04.028
Pegoli, A., Wifling, D., Gruber, C.G., She, X., Hübner, H., Bernhardt, G.,... Keller, M. (2019). Conjugation of Short Peptides to Dibenzodiazepinone-Type Muscarinic Acetylcholine Receptor Ligands Determines M2R Selectivity. Journal of Medicinal Chemistry, 62(11), 5358-5369. https://dx.doi.org/10.1021/acs.jmedchem.8b01967
Schwalbe, T., Hübner, H., & Gmeiner, P. (2019). Development of covalent antagonists for beta 1-and beta 2-adrenergic receptors. Bioorganic & Medicinal Chemistry, 27(13), 2959-2971. https://dx.doi.org/10.1016/j.bmc.2019.05.034
Stanek, M., Picard, L.P., Schmidt, M., Kaindl, J., Hübner, H., Bouvier, M.,... Gmeiner, P. (2019). Hybridization of β-Adrenergic Agonists and Antagonists Confers G Protein Bias. Journal of Medicinal Chemistry, 62(10), 5111-5131. https://dx.doi.org/10.1021/acs.jmedchem.9b00349
Sommer, T., Dlugash, G., Hübner, H., Gmeiner, P., & Pischetsrieder, M. (2019). Monitoring of the dopamine D2 receptor agonists hordenine and N-methyltyramine during the brewing process and in commercial beer samples. Food Chemistry, 276, 745-753. https://dx.doi.org/10.1016/j.foodchem.2018.10.067
Kling, R., Burchardt, C., Einsiedel, J., Hübner, H., & Gmeiner, P. (2019). Structure-based exploration of an allosteric binding pocket in the NTS1 receptor using bitopic NT(8-13) derivatives and molecular dynamics simulations. Journal of Molecular Modeling, 25(7). https://dx.doi.org/10.1007/s00894-019-4064-x
Nebel, N., Strauch, B., Maschauer, S., Lasch, R., Rampp, H., Fehler, S.,... Prante, O. (2017). 18F]Fluorophenylazocarboxylates: Design and Synthesis of Potential Radioligands for Dopamine D3 and μ-Opioid Receptor. ACS Omega, 2(12), 8649-8659. https://dx.doi.org/10.1021/acsomega.7b01374
Nebel, N., Strauch, B., Maschauer, S., Lasch, R., Rampp, H., Fehler, S.,... Prante, O. (2017). [18F]Fluorophenylazocarboxylates: Design and Synthesis of Potential Radioligands for Dopamine D3 and μ‑Opioid Receptor. ACS Omega, 2, 8649-8659. https://dx.doi.org/10.1021/acsomega.7b01374
Männel, B., Hübner, H., Möller, D., & Gmeiner, P. (2017). beta-Arrestin biased dopamine D2 receptor partial agonists: Synthesis and pharmacological evaluation. Bioorganic & Medicinal Chemistry, 25(20), 5613-5628. https://dx.doi.org/10.1016/j.bmc.2017.08.037
Stößel, A., Brox, R., Purkayastha, N., Hübner, H., Hocke, C., Prante, O., & Gmeiner, P. (2017). Development of molecular tools based on the dopamine D3 receptor ligand FAUC 329 showing inhibiting effects on drug and food maintained behavior. Bioorganic & Medicinal Chemistry, 25(13), 3491-3499. https://dx.doi.org/10.1016/j.bmc.2017.04.036

Last updated on 2016-05-05 at 05:06