Lehrstuhl für Pharmazeutische Chemie

Adresse:
Nikolaus-Fiebiger-Str. 10
91058 Erlangen



Untergeordnete Organisationseinheiten

Professur für Pharmazeutische Chemie
Professur für Pharmazeutische Chemie


Publikationen (Download BibTeX)

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Möller, D., Banerjee, A., Uzuneser, T., Skultety, M., Huth, T., Plouffe, B.,... Gmeiner, P. (2017). Discovery of G Protein-Biased Dopaminergics with a Pyrazolo[1,5-a]pyridine Substructure. Journal of Medicinal Chemistry, 60(7), 2908-2929. https://dx.doi.org/10.1021/acs.jmedchem.6b01857
Sommer, T., Hübner, H., El Kerdawy, A., Gmeiner, P., Pischetsrieder, M., & Clark, T. (2017). Identification of the Beer Component Hordenine as Food-Derived Dopamine D2 Receptor Agonist by Virtual Screening a 3D Compound Database. Scientific Reports, 7, 44201. https://dx.doi.org/10.1038/srep44201
She, X., Pegoli, A., Mayr, J., Hübner, H., Bernhardt, G., Gmeiner, P., & Keller, M. (2017). Heterodimerization of dibenzodiazepinone-type muscarinic acetylcholine receptor ligands leads to increased M2R affinity and selectivity. ACS Omega, 2(10), 6741-6754. https://dx.doi.org/10.1021/acsomega.7b01085
Maschauer, S., Einsiedel, J., Reich, D., Hübner, H., Gmeiner, P., Wester, H.J.,... Notni, J. (2017). Theranostic Value of Multimers: Lessons Learned from Trimerization of Neurotensin Receptor Ligands and Other Targeting Vectors. Pharmaceuticals, 10(1), 29. https://dx.doi.org/10.3390/ph10010029
Fröhlich, T., Reiter, C., Ibrahim, M.M., Beutel, J., Hutterer, C., Zeitträger, I.,... Tsogoeva, S. (2017). Synthesis of Novel Hybrids of Quinazoline and Artemisinin with High Activities against Plasmodium falciparum, Human Cytomegalovirus, and Leukemia Cells. ACS Omega, 2(6), 2422-2431. https://dx.doi.org/10.1021/acsomega.7b00310
Nebel, N., Strauch, B., Maschauer, S., Lasch, R., Rampp, H., Fehler, S.,... Prante, O. (2017). 18F]Fluorophenylazocarboxylates: Design and Synthesis of Potential Radioligands for Dopamine D3 and μ-Opioid Receptor. ACS Omega, 2(12), 8649-8659. https://dx.doi.org/10.1021/acsomega.7b01374
Stößel, A., Brox, R., Purkayastha, N., Hübner, H., Hocke, C., Prante, O., & Gmeiner, P. (2017). Development of molecular tools based on the dopamine D3 receptor ligand FAUC 329 showing inhibiting effects on drug and food maintained behavior. Bioorganic & Medicinal Chemistry, 25(13), 3491-3499. https://dx.doi.org/10.1016/j.bmc.2017.04.036
Simeth, N.A., Bause, M., Dobmeier, M., Kling, R., Lachmann, D., Hübner, H.,... Koenig, B. (2017). NTS2-selective neurotensin mimetics with tetrahydrofuran amino acids. Bioorganic & Medicinal Chemistry, 25(1), 350-359. https://dx.doi.org/10.1016/j.bmc.2016.10.039
Nebel, N., Strauch, B., Maschauer, S., Lasch, R., Rampp, H., Fehler, S.,... Prante, O. (2017). [18F]Fluorophenylazocarboxylates: Design and Synthesis of Potential Radioligands for Dopamine D3 and μ‑Opioid Receptor. ACS Omega, 2, 8649-8659. https://dx.doi.org/10.1021/acsomega.7b01374
Tabor, A., Möller, D., Hübner, H., Kornhuber, J., & Gmeiner, P. (2017). Visualization of ligand-induced dopamine D2S and D2L receptor internalization by TIRF microscopy. Scientific Reports, 7, 10894. https://dx.doi.org/10.1038/s41598-017-11436-1
Milanos, L., Saleh, N., Kling, R., Kaindl, J., Tschammer, N., & Clark, T. (2016). Identification of Two Distinct Sites for Antagonist and Biased Agonist Binding to the Human Chemokine Receptor CXCR3. Angewandte Chemie-International Edition, 55(49), 15277-15281. https://dx.doi.org/10.1002/anie.201607831
Tabor, A., Weisenburger, S., Banerjee, A., Purkayastha, N., Kaindl, J., Hübner, H.,... Gmeiner, P. (2016). Visualization and ligand-induced modulation of dopamine receptor dimerization at the single molecule level. Scientific Reports, 6, 33233. https://dx.doi.org/10.1038/srep33233
Manglik, A., Lin, H., Aryal, D.K., Mccorvy, J.D., Dengler, D., Corder, G.,... Shoichet, B.K. (2016). Structure-based discovery of opioid analgesics with reduced side effects. Nature, 537(7619), 185-190. https://dx.doi.org/10.1038/nature19112
Ludwig, J., Ulm, N., Pröschel, M., Sticht, H., Sonnewald, U., & Eichler, J. (2016). CHARACTERIZATION OF THE SPYTAG - SPY-CATCHER INTERACTION. Journal of Peptide Science, 22, S66-S66.
Naporra, F., Gobleder, S., Wittmann, H.-J., Spindler, J., Bodensteiner, M., Bernhardt, G.,... Strasser, A. (2016). Dibenzo[b,f][1,4]oxazepines and dibenzo[b,e]oxepines: Influence of the chlorine substitution pattern on the pharmacology at the H1R, H4R, 5-HT2AR and other selected GPCRs. Pharmacological research, 113, 610-625. https://dx.doi.org/10.1016/j.phrs.2016.09.042
Röhrig, W., Waibel, R., Perlwitz, C., Pischetsrieder, M., & Hoch, T. (2016). Identification of the oleic acide ethanolamide (OEA) isomer cis-vaccenic acid ethanolamide (VEA) as a highly abundant 18:1 fatty acid ethanolamide in blood plasma from rats and humans. Analytical and Bioanalytical Chemistry, 408(22), 6141-6151. https://dx.doi.org/10.1007/s00216-016-9720-8
Weichert, D., Stanek, M., Hübner, H., & Gmeiner, P. (2016). Structure-guided development of dual ß2 adrenergic/dopamine D-2 receptor agonists. Bioorganic & Medicinal Chemistry, 24, 2641-2653. https://dx.doi.org/10.1016/j.bmc.2016.04.028
Maia de Pádua, R., Meitinger, N., Hennemann, M., Schebitz, P., Waibel, R., Löber, S.,... Kreis, W. (2016). Spontaneous butenolide ring formation of pregnane-21-O-malonyl hemiesters under mild reaction conditions is facilitated by the 14β-hydroxy group present in all natural cardenolides. Tetrahedron, 72, 4556-4563. https://dx.doi.org/10.1016/j.tet.2016.06.024
Kling, R., Plomer, M., Lang, C., Banerjee, A., Hübner, H., & Gmeiner, P. (2016). Development of Covalent Ligand-Receptor Pairs to Study the Binding Properties of Nonpeptidic Neurotensin Receptor 1 Antagonists. ACS chemical biology, 11(4), 869-875. https://dx.doi.org/10.1021/acschembio.5b00965
Lampros, M., Brox, R., Frank, T., Poklukar, G., Palmisano, R., Waibel, R.,... Tschammer, N. (2016). Discovery and Characterization of Biased Allosteric Agonists of the Chemokine Receptor CXCR3. Journal of medicinal chemistry, 59(5), 2222-43. https://dx.doi.org/10.1021/acs.jmedchem.5b01965

Zuletzt aktualisiert 2019-24-04 um 10:21